Cesare Gennari - Publications#

H index (Scopus): 48 (26/09/2024)
Total citations (Scopus): 8.780 (26/09/2024)

Selected Publications

1) Amine-Carbamate Self-Immolative Spacers Counterintuitively Release 3° Alcohol at Much Faster Rates than 1° Alcohol Payloads
M. Mason, L. Bisbal Lopez, F. Bashiri, A. Herrero, A. Baron, R. Bucci, L. Pignataro, C. Gennari, A. Dal Corso
ChemBioChem 2024, DOI: 10.1002/cbic.202400174

2) RGD Cyclopeptide Equipped with a Lysine-Engaging Salicylaldehyde Showing Enhanced Integrin Affinity and Cell Detachment Potency
G. Sacco, D. Arosio, M. Paolillo, A. Gloger, J. Scheuermann, L. Pignataro, L. Belvisi, A. Dal Corso, C. Gennari
Chem. Eur. J. 2023, 29, e202203768

3) Fast Cyclization of a Proline-Derived Self-Immolative Spacer Improves the Efficacy of Carbamate Prodrugs
Dal Corso, A.; Borlandelli, V.; Corno, C.; Perego, P.; Belvisi, L.; Pignataro, L.; Gennari, C.
Angew. Chem. Int. Ed. 2020, 59, 4176-4181; DOI: 10.1002/anie.201916394

4) Multimeric Presentation of RGD Peptidomimetics Enhances Integrin Binding and Tumor Cell Uptake
Pina, A.; Kadri, M.; Arosio, D.; Dal Corso, A.; Coll, J.-L.; Gennari, C.; Boturyn, D.
Chemistry - A European Journal 2020, 26, 7492-7496; DOI: 10.1002/chem.202001115

5) Innovative linker strategies for tumor-targeted drug conjugates
Dal Corso, A.; Pignataro, L.; Belvisi, L.; Gennari, C.
Chemistry - A European Journal 2019, 25, 14740-14757; DOI: 10.1002/chem.201903127

6) Neutrophil Elastase Promotes Linker Cleavage and Paclitaxel Release from an Integrin-Targeted Conjugate
Raposo Moreira Dias, A.; Pina, A.; Dean, A.; Lerchen, H.-G.; Caruso, M.; Gasparri, F.; Fraietta, I.; Troiani, S.; Arosio, D.; Belvisi, L.; Pignataro, L.; Dal Corso, A.; Gennari, C.
Chemistry - A European Journal 2019, 25, 1696-1700; DOI: 10.1002/chem.201805447

7) Efficient Synthesis of Amines by Iron-Catalyzed C=N Transfer Hydrogenation and C=O Reductive Amination
Vailati Facchini, S.; Cettolin, M.; Bai, X.; Casamassima, G.; Pignataro, L.; Gennari, C.; Piarulli, U.
Adv. Synth. Catal. 2018, 360, 1054-1059; DOI 10.1002/adsc.201701316

8) Multivalency Increases the Binding Strength of RGD Peptidomimetic-Paclitaxel Conjugates to Integrin aVb3
Raposo Moreira Dias, A.; Pina, A.; Dal Corso, A.; Arosio, D.; Belvisi, L.; Pignataro, L.; Caruso, M.; Gennari, C.
Chemistry - A European Journal 2017, 23, 14410-14415; DOI: 10.1002/chem.201703093

9) Tumor Targeting with an isoDGR-Drug Conjugate
Zanella, S.; Angerani, S.; Pina, A.; López Rivas, P.; Giannini, C.; Panzeri, S.; Arosio, D.; Caruso, M.; Gasparri, F.; Fraietta, I.; Albanese, C.; Marsiglio, A.; Pignataro, L.; Belvisi, L.; Piarulli, U.; Gennari, C.
Chemistry - A European Journal 2017, 23, 7910-7914; DOI: 10.1002/chem.201701844

10) Asymmetric Transfer Hydrogenation of Ketones with modified Grubbs Metathesis Catalysts: On the Way to a Tandem Process
Renom-Carrasco, M.; Gajewski, P.; Pignataro, L.; de Vries, J. G.; Piarulli, U.; Gennari, C.; Lefort, L.
Adv. Synth. Catal. 2016, 358, 515-519; DOI: 10.1002/adsc.201500933